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NO-1886 upregulates ATP binding cassette transporter A1 and inhibits diet-induced atherosclerosis in Chinese Bama minipigs

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成果类型:
期刊论文
作者:
Zhang, Chi;Yin, Weidong*;Liao, Duanfang;Huang, Liang;Tang, Chaoke;...
通讯作者:
Yin, Weidong
作者机构:
[Yin, Weidong] Nanhua Univ, Sch Med, Inst Cardiovasc Res, Hengyang 421001, Hunan, Peoples R China.
Nanhua Univ, Sch Life Sci & Technol, Dept Biochem & Mol Biol, Hengyang 421001, Hunan, Peoples R China.
Nanhua Univ, Sch Med, Funct Lab Ctr, Hengyang 421001, Hunan, Peoples R China.
Nanhua Univ, Inst Pharm & Pharmacol, Hengyang 421001, Hunan, Peoples R China.
Nanhua Univ, Sch Med, Dept Operat Surg, Hengyang 421001, Hunan, Peoples R China.
通讯机构:
[Yin, Weidong] N
Nanhua Univ, Sch Med, Inst Cardiovasc Res, Hengyang 421001, Hunan, Peoples R China.
语种:
英文
关键词:
liver X receptor alpha;scavenger receptor class B type I;[4-(4-bromo-2-cyano-phenylcarbamoyl)-benzyl] phosphonic;acid diethyl ester
关键词(中文):
动脉粥样硬化;胆固醇
期刊:
Journal of Lipid Research
ISSN:
0022-2275
年:
2006
卷:
47
期:
9
页码:
2055-2063
机构署名:
本校为第一且通讯机构
院系归属:
化学化工学院
医学院
药学与生物科学学院
摘要:
It is widely believed that high density lipoprotein-cholesterol (HDL-C) functions to transport cholesterol from peripheral cells to the liver by reverse cholesterol transport (RCT), a pathway that may protect against atherosclerosis by clearing excess cholesterol from arterial cells. A cellular ATP binding cassette transporter called ABCA1 mediates the first step of RCT. NO-1886 has been proven to be highly effective at increasing HDL-C and reducing atherosclerosis. However, the mechanism of atherosclerosis inhibition for NO-1886 is not fully u...

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