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Disulfiram: A novel repurposed drug for cancer therapy

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成果类型:
期刊论文
作者:
Zeng, Min;Wu, Baibei;Wei, Wenjie;Jiang, Zihan;Li, Peiqiang;...
作者机构:
[Zeng, Min; Jiang, Zihan; Li, Peiqiang; Quan, Yuanting] Department of Biochemistry and Molecular Biology, School of Basic Medicine, Hengyang Medical School, University of South China, Hengyang, Hunan 421001, China
[Wu, Baibei] The Key Laboratory of Ecological Environment and Critical Human Diseases Prevention of Hunan Province Department of Education, Hengyang Medical School, University of South China, Hengyang, Hunan 421001, China
[Wei, Wenjie] Institute of Biochemistry of Hengyang Medical School, University of South China, Hengyang, Hunan 421001, China.
[Hu, Xiaobo] Department of Biochemistry and Molecular Biology, School of Basic Medicine, Hengyang Medical School, University of South China, Hengyang, Hunan 421001, China<&wdkj&>The Key Laboratory of Ecological Environment and Critical Human Diseases Prevention of Hunan Province Department of Education, Hengyang Medical School, University of South China, Hengyang, Hunan 421001, China
语种:
英文
关键词:
Disulfiram;Aldehyde dehydrogenase;Reactive oxygen species;Proteasome activity;Cancer stem cells;Drug resistance
期刊:
中华医学杂志(英文版)
ISSN:
0366-6999
年:
2024
机构署名:
本校为第一机构
院系归属:
化学化工学院
摘要:
Cancer is a major global health issue. Effective therapeutic strategies can prolong patients' survival and reduce the costs of treatment. Drug repurposing, which identifies new therapeutic uses for approved drugs, is a promising approach with the advantages of reducing research costs, shortening development time, and increasing efficiency and safety. Disulfiram (DSF), an Food and Drug Administration (FDA)-approved drug used to treat chronic alcoholism, has a great potential as an anticancer drug by targeting diverse human malignancies. Several ...

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